SANTO PREVITI

Work

Vrije Universiteit Brussel

Belgium

Publications

The Role of Nutraceuticals in Age-Related Ocular Diseases

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Molecules

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The Role of Nutraceuticals in Age-Related Ocular Diseases

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Molecules

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Inhibitors of Proteases: A Well-Grounded Strategy in Drug Development

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Molecules

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A Second Opportunity for the Peptide-Based Analogues with γ-Lactam at the P1 Position: Human Cathepsin S Inhibition

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Pharmaceuticals

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Inhibitors of Proteases: A Well-Grounded Strategy in Drug Development

Published by

Molecules

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Synthesis and Combination Studies of Novel Dipeptide Nitriles with Curcumin for a Potent Synergistic Action Against Rhodesain, Cysteine Protease of Trypanosoma brucei rhodesiense

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Pharmaceuticals

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Synthesis and Combination Studies of Novel Dipeptide Nitriles with Curcumin for a Potent Synergistic Action Against Rhodesain, Cysteine Protease of <i>Trypanosoma brucei rhodesiense</i>

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Pharmaceuticals

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Identification of constrained peptidomimetics carrying a Michael acceptor warhead as antitrypanosomal agents

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European Journal of Medicinal Chemistry

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Identification of constrained peptidomimetics carrying a Michael acceptor warhead as antitrypanosomal agents

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European Journal of Medicinal Chemistry

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Design and Synthesis of <SUP>68</SUP>Ga-Labeled Peptide-Based Heterodimers for Dual Targeting of NTS<sub>1</sub> and GRPR

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ChemMedChem

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N-Terminal Stabilization of Radiolabeled Neurotensin Analogues for Improved Tumor Uptake

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Journal of Medicinal Chemistry

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The Role of Nutraceuticals in Chemoprevention and their Therapeutic Effects when used in Combination with Synthetic Drugs

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Current Medicinal Chemistry

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Drug Combination Studies of Isoquinolinone AM12 with Curcumin or Quercetin: A New Combination Strategy to Synergistically Inhibit 20S Proteasome

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International Journal of Molecular Sciences

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Drug Combination Studies of Isoquinolinone AM12 with Curcumin or Quercetin: A New Combination Strategy to Synergistically Inhibit 20S Proteasome

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International Journal of Molecular Sciences

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Drug Combination Studies of Isoquinolinone AM12 with Curcumin or Quercetin: A New Combination Strategy to Synergistically Inhibit 20S Proteasome

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International Journal of Molecular Sciences

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Design, Synthesis, and In Vitro Characterization of Proteolytically-Stable Opioid-Neurotensin Hybrid Peptidomimetics

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ACS Pharmacology & Translational Science

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Design, Synthesis, and In Vitro Characterization of ProteolyticallyStable Opioid-Neurotensin Hybrid Peptidomimetics

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ACS pharmacology & translational science

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Identification of Dual Inhibitors Targeting Main Protease (Mpro) and Cathepsin L as Potential Anti-SARS-CoV-2 Agents

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ACS Medicinal Chemistry Letters

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Identification of Dual Inhibitors Targeting Main Protease (M<SUP>pro</SUP>) and Cathepsin L as Potential Anti-SARS-CoV-2 Agents

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ACS Medicinal Chemistry Letters

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Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria

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International Journal of Molecular Sciences

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Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria

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International Journal of Molecular Sciences

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The Inhibition of NS2B/NS3 Protease: A New Therapeutic Opportunity to Treat Dengue and Zika Virus Infection

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International Journal of Molecular Sciences

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The Inhibition of NS2B/NS3 Protease: A New Therapeutic Opportunity to Treat Dengue and Zika Virus Infection

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International Journal of Molecular Sciences

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Rational design of NT-PSMA heterobivalent probes for prostate cancer theranostics

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RSC Medicinal Chemistry

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Opening the amino acid toolbox for peptide-based NTS2-selective ligands as promising lead compounds for pain management

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Journal of Peptide Science

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Influence of amino acid size at the P3 position of N-Cbz-tripeptide Michael acceptors targeting falcipain-2 and rhodesain for the treatment of malaria and human african trypanosomiasis

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Bioorganic Chemistry

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Influence of amino acid size at the P3 position of N-Cbz-tripeptide Michael acceptors targeting falcipain-2 and rhodesain for the treatment of malaria and human african trypanosomiasis

Published by

Bioorganic Chemistry

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Opening the amino acid toolbox for peptide‐based NTS2‐selective ligands as promising lead compounds for pain management

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Journal of Peptide Science

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Opening the amino acid toolbox for peptide-based NTS2-selective ligands as promising lead compounds for pain management

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Journal of Peptide Science

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Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense

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International Journal of Molecular Sciences

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Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of <i>Trypanosoma brucei rhodesiense</i>

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International Journal of Molecular Sciences

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Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of <i>Trypanosoma brucei rhodesiense</i>

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International Journal of Molecular Sciences

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Monoclonal Antibodies: The Greatest Resource to Treat Multiple Myeloma

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International Journal of Molecular Sciences

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Monoclonal Antibodies: The Greatest Resource to Treat Multiple Myeloma

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International Journal of Molecular Sciences

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Monoclonal Antibodies: The Greatest Resource to Treat Multiple Myeloma

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International Journal of Molecular Sciences

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Structure-based lead optimization of peptide-based vinyl methyl ketones as SARS-CoV-2 main protease inhibitors

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European Journal of Medicinal Chemistry

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Structure-based lead optimization of peptide-based vinyl methyl ketones as SARS-CoV-2 main protease inhibitors

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European Journal of Medicinal Chemistry

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Development of biased/selective OP-NT hybrids for pain treatment

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23rd GFPP meeting, Fournols Auvergne, France, 17/09/23

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conference-poster

Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of <i>Trypanosoma brucei rhodesiense</i>

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International Journal of Molecular Sciences

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Dual Inhibition of Parasitic Targets: A Valuable Strategy to Treat Malaria and Neglected Tropical Diseases

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Current Medicinal Chemistry

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Drug Combination Studies of the Dipeptide Nitrile CD24 with Curcumin: A New Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense

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International Journal of Molecular Sciences

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Development of isoquinolinone derivatives as immunoproteasome inhibitors

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Bioorganic & Medicinal Chemistry Letters

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Development of Urea-Bond-Containing Michael Acceptors as Antitrypanosomal Agents Targeting Rhodesain

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ACS Medicinal Chemistry Letters

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Development of Reduced Peptide Bond Pseudopeptide Michael Acceptors for the Treatment of Human African Trypanosomiasis

Published by

Molecules

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Development of Reduced Peptide Bond Pseudopeptide Michael Acceptors for the Treatment of Human African Trypanosomiasis

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Molecules

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Design and NMR conformational analysis in solution of β5i-selective inhibitors of immunoproteasome

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Journal of Molecular Structure

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Lead Discovery of SARS-CoV-2 Main Protease Inhibitors through Covalent Docking-Based Virtual Screening

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Journal of Chemical Information and Modeling

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Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal Structure †

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Journal of medicinal chemistry

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Falcipain-2 and Falcipain-3 Inhibitors as Promising Antimalarial Agents

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Current Medicinal Chemistry

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Drug Synergism: Studies of Combination of RK-52 and Curcumin against Rhodesain of Trypanosoma brucei rhodesiense

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ACS Medicinal Chemistry Letters

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Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure-Activity Relationship Studies

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Journal of medicinal chemistry

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Design and NMR conformational analysis in solution of β5i-selective inhibitors of immunoproteasome

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Journal of Molecular Structure

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Silicon-Containing Neurotensin Analogues as Radiopharmaceuticals for NTS1-Positive Tumors Imaging

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Bioconjugate Chemistry

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Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment

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ChemMedChem

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Insightful Backbone Modifications Preventing Proteolytic Degradation of Neurotensin Analogs Improve NT S1-Induced Protective Hypothermia.

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Frontiers in Chemistry

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Drug Synergism: Studies of Combination of RK-52 and Curcumin against Rhodesain of Trypanosoma brucei rhodesiense

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ACS Medicinal Chemistry Letters

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Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense

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ChemMedChem

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Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense

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Natural Product Research

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Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis

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Journal of Medicinal Chemistry

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Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis

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Journal of Medicinal Chemistry

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Design and evaluation of non-carboxylate 5-arylidene-2-thioxo-4-imidazolidinones as novel non-competitive inhibitors of protein tyrosine phosphatase 1B

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Bioorganic Chemistry

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Evaluation of curcumin irreversibility

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Natural Product Research

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Identification of 2-thioxoimidazolidin-4-one derivatives as novel noncovalent proteasome and immunoproteasome inhibitors

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Bioorganic & Medicinal Chemistry Letters

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Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs)

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Journal of Medicinal Chemistry

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Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs)

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Journal of Medicinal Chemistry

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Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors

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Journal of Enzyme Inhibition and Medicinal Chemistry

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The Inhibition of Cysteine Proteases Rhodesain and TbCatB: A Valuable Approach to Treat Human African Trypanosomiasis

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Mini-Reviews in Medicinal Chemistry

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Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agents

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Bioorganic & Medicinal Chemistry Letters

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Immunoproteasome-Selective Inhibitors: A Promising Strategy to Treat Hematologic Malignancies, Autoimmune and Inflammatory Diseases

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Current Medicinal Chemistry

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Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation

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Bioorganic and Medicinal Chemistry

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